2. Strategies based on transforms I.
Selection of disconnections
|
2.1. C-X disconnections of monofunctional compounds
2.2. C-X disconnections of difunctional compounds (1, n)
2.3. C-C disconnections of monofunctional compounds
2.4. C-C disconnections of difunctional compounds (1, n)
2.5. Aromatic Compound Disconnections |
4. Strategy based on functional groups II. Protective groups in Organic synthesis
|
4.1. Description of the protecting groups.
4.2. Sensitive to acid, basic, fluoride, oxidizing agents and reducing agents.
4.3. Selection of protecting groups |
| 6. Strategy based on stereochemical |
6.1. Description of stereochemistry. Chirality and descriptors. Topicity
6.2. Stereochemistry of chemical reactions. Product selectivity. Simple and induced diastereoselectivity.
|
Experimental Section. The synthetic milestone of design and discovery of organic compounds with
therapeutic applications. |
4 sessions |
